Description
Diferelin (Triptorelin) Powder 0.1 mg Injections №7
Ingredients:
Active ingredient: Triptorelin acetate. Inactive ingredients may include mannitol and acetic acid for pH adjustment.
Mechanism of Action:
Diferelin (triptorelin) acts by continuously stimulating the pituitary gland to produce and release gonadotropins, ultimately leading to a decrease in testosterone levels in men and estrogen levels in women. This mechanism is crucial in the treatment of hormone-sensitive conditions.
Pharmacological Properties:
Diferelin belongs to the class of gonadotropin-releasing hormone (GnRH) agonists. It exerts its effects by desensitizing the GnRH receptors in the pituitary gland, leading to the suppression of gonadotropin secretion.
Indications for Use:
- Treatment of advanced prostate cancer
- Management of endometriosis
- Control of central precocious puberty
Contraindications:
Do not use Diferelin if:
- Allergic to triptorelin or any components
- Pregnant
- Breastfeeding
Side Effects:
Common side effects of Diferelin may include hot flashes, decreased libido, fatigue, and injection site reactions. Patients should consult their healthcare provider for a full list of possible adverse effects.
Usage Instructions:
Usual Dosage: 0.1 mg injected subcutaneously once a day. Patients should follow the healthcare provider’s instructions for the correct administration of the injections. Store at room temperature away from moisture and heat.
Benefits Compared to Analogues:
Comparative studies have shown that Diferelin exhibits similar efficacy to other GnRH agonists but with potentially fewer side effects, making it a preferred choice in clinical practice.
Suitable Patient Groups:
Diferelin is suitable for adult patients including the elderly. Pediatric use should be determined by a healthcare provider based on individual considerations.
Storage Conditions and Shelf Life:
Store Diferelin as per the instructions provided in the packaging. Check the expiration date and do not use the product beyond the stated shelf life.
Packaging Description:
Diferelin is available in packs containing 7 powder injections of 0.1 mg strength each. The packaging should be intact and undamaged before use.